Preparation of enantioenriched α-bromo acids incorporating diverse functionality

Andrew J. Souers, Stephan C Schuerer, Heemun Kwack, Alex A. Virgilio, Jonathan A. Ellman

Research output: Contribution to journalArticle

15 Citations (Scopus)

Abstract

A number of enantioenriched α-bromo acids with diverse side chain functionality have been synthesized in one step from their corresponding protected α-amino acids. Good yields and excellent enantiopurities were observed for all substrates examined.

Original languageEnglish
Pages (from-to)583-585
Number of pages3
JournalSynthesis
Issue number4
StatePublished - Jan 1 1999
Externally publishedYes

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Amino acids
Amino Acids
Acids
Substrates

Keywords

  • α-amino acids
  • α-bromo acids
  • Acid labile side chain protecting groups

ASJC Scopus subject areas

  • Organic Chemistry

Cite this

Souers, A. J., Schuerer, S. C., Kwack, H., Virgilio, A. A., & Ellman, J. A. (1999). Preparation of enantioenriched α-bromo acids incorporating diverse functionality. Synthesis, (4), 583-585.

Preparation of enantioenriched α-bromo acids incorporating diverse functionality. / Souers, Andrew J.; Schuerer, Stephan C; Kwack, Heemun; Virgilio, Alex A.; Ellman, Jonathan A.

In: Synthesis, No. 4, 01.01.1999, p. 583-585.

Research output: Contribution to journalArticle

Souers, AJ, Schuerer, SC, Kwack, H, Virgilio, AA & Ellman, JA 1999, 'Preparation of enantioenriched α-bromo acids incorporating diverse functionality', Synthesis, no. 4, pp. 583-585.
Souers AJ, Schuerer SC, Kwack H, Virgilio AA, Ellman JA. Preparation of enantioenriched α-bromo acids incorporating diverse functionality. Synthesis. 1999 Jan 1;(4):583-585.
Souers, Andrew J. ; Schuerer, Stephan C ; Kwack, Heemun ; Virgilio, Alex A. ; Ellman, Jonathan A. / Preparation of enantioenriched α-bromo acids incorporating diverse functionality. In: Synthesis. 1999 ; No. 4. pp. 583-585.
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